Activity [%Ctr] | FFAR2 | FFAR3 | GPR119 | GPR120 | GPR55 | GPR142 | GLP1R | PPARγ | PPARα |
---|---|---|---|---|---|---|---|---|---|
Assay | Calcium flux | cAMP | β-Arrestin | β-Arrestin | β-Arrestin | β-Arrestin | β-Arrestin | NHR Protein Interaction | NHR Protein Interaction |
CPL207280 | −1 | 28.5 | 9.1 | 0.5 | 6.3 | 8.5 | −2.6 | 1.2 | 0.9 |
TAK-875 | 9.1 | 22.8 | 7.3 | 6 | 14.8 | −13.4 | −1.5 | 4.1 | 8.7 |