Understanding the structure-activity relationship of the human ether-a-go-go-related gene cardiac K+ channel. A model for bad behavior

J Med Chem. 2003 May 22;46(11):2017-22. doi: 10.1021/jm0205651.
No abstract available

Publication types

  • Review

MeSH terms

  • Cation Transport Proteins*
  • DNA-Binding Proteins*
  • Drug-Related Side Effects and Adverse Reactions*
  • ERG1 Potassium Channel
  • Ether-A-Go-Go Potassium Channels
  • Humans
  • Long QT Syndrome / chemically induced
  • Models, Molecular
  • Pharmaceutical Preparations / chemistry*
  • Potassium Channels / chemistry
  • Potassium Channels / drug effects*
  • Potassium Channels, Voltage-Gated*
  • Structure-Activity Relationship
  • Torsades de Pointes / chemically induced
  • Trans-Activators*
  • Transcriptional Regulator ERG

Substances

  • Cation Transport Proteins
  • DNA-Binding Proteins
  • ERG protein, human
  • ERG1 Potassium Channel
  • Ether-A-Go-Go Potassium Channels
  • KCNH2 protein, human
  • KCNH6 protein, human
  • Pharmaceutical Preparations
  • Potassium Channels
  • Potassium Channels, Voltage-Gated
  • Trans-Activators
  • Transcriptional Regulator ERG