Ligand-selective signaling and high-content screening for GPCR drugs

Drug Discov Today. 2003 Dec 15;8(24):1108-9. doi: 10.1016/s1359-6446(03)02897-6.
No abstract available

Publication types

  • Comment

MeSH terms

  • Drug Design
  • Drug Evaluation, Preclinical
  • Humans
  • Ligands
  • Molecular Conformation
  • Quinuclidines / pharmacology
  • Receptor, Muscarinic M1 / agonists
  • Receptors, G-Protein-Coupled / agonists
  • Receptors, G-Protein-Coupled / drug effects*
  • Receptors, G-Protein-Coupled / metabolism
  • Receptors, G-Protein-Coupled / physiology
  • Signal Transduction
  • Thiophenes*

Substances

  • Ligands
  • Quinuclidines
  • Receptor, Muscarinic M1
  • Receptors, G-Protein-Coupled
  • Thiophenes
  • cevimeline