Computational modeling to accelerate the identification of substrates and inhibitors for transporters that affect drug disposition

Clin Pharmacol Ther. 2012 Nov;92(5):661-5. doi: 10.1038/clpt.2012.164. Epub 2012 Sep 26.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Computational Biology*
  • Drug Interactions
  • Drug-Related Side Effects and Adverse Reactions
  • Humans
  • Ligands
  • Membrane Transport Proteins / chemistry
  • Membrane Transport Proteins / metabolism*
  • Models, Biological*
  • Pharmaceutical Preparations / metabolism*
  • Structure-Activity Relationship

Substances

  • Ligands
  • Membrane Transport Proteins
  • Pharmaceutical Preparations