Most drugs are bound to human serum albumin (HSA) via a few high affinity binding sites
and several sites of much lower affinity. There is now increasing evidence that the actual …

The interaction of several β-carbolines with specific [ 3 H]-flunitrazepam binding to
benzodiazepine receptors in rat brain membranes was investigated. Out of the investigated …

β-Carbolines have been recently proposed as candidates for the unknown endogenous
ligand of the benzodiazepine receptor. Out of the β-carboline derivatives already found in the …

Harmane and other related β-carbolines are putative endogenous ligands of the benzodiazepine
receptor. Since the compounds are potent convulsants they may have agonist activities …

The interaction of warfarin and dicoumarol with tryptophan- and tyrosine-modified human
serum albumin derivatives was investigated by equilibrium dialysis and circular dichroism …

Penicillins are thought to be GABA receptor antagonists. In order to determine the affinities of
various penicillin derivatives for the GABA receptor, their potencies as inhibitors of specific [ …

The interaction of L-tryptophan and four benzodiazepine derivatives with tyrosine-modified
human serum albumin was investigated by equilibrium dialysis and circular dichroism …

Using d- and l-oxazepam hemisuccinate (RV 1208 and RV 1210), the stereospecificity of
binding of benzodiazepines to human serum albumin was investigated. The interactions of the …

The binding of suramin to bovine and human serum albumin was investigated by gel filtration
and spectroscopic measurements. Besides some low-affinity binding sites suramin has, on …

The interaction of seven penicillin derivatives with specific [ 3 H]flunitrazepam binding to
benzodiazepine receptors was investigated. The affinities of the penicillins for benzodiazepine …