Fast Forward

Molecular Pharmacology Fast Forward contains papers in manuscript form that have been accepted and published in Molecular Pharmacology but have not been copyedited and have not been assigned to an issue of the journal. Copyediting may lead to some differences between the Fast Forward version and the final version. There may also be differences in the quality of the graphics. The publication date appears below each title followed by the article's unique Digital Object Identifier (DOI).

Articles

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Pyrimidinyl Biphenylureas Act as Allosteric Modulators to activate Cannabinoid Receptor 1 and initiate β-Arrestin-dependent Responses
Caitlin A.D. Jagla, Caitlin E. Scott, Yaliang Tang, Changjiang Qiao, Gabriel E. Mateo-Semidey, Guillermo A. Yudowski, Dai Lu and Debra A. Kendall

Molecular Pharmacology October 15, 2018, mol.118.112854; DOI: https://doi.org/10.1124/mol.118.112854
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Involvement of 5-HT_1A and 5-HT_2A receptors but not α₂-adrenoceptors in the acute electrophysiological effects of cariprazine in the rat brain in vivo
Anna Herman, Mostafa El Mansari, Nika Adham, Bela Kiss, Bence Farkas and Pierre Blier

Molecular Pharmacology October 15, 2018, mol.118.113290; DOI: https://doi.org/10.1124/mol.118.113290
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Physicochemical solubility of and biological sensitivity to long-chain alcohols determine the cutoff chain length in biological activity
Atsushi Matsumoto and Yukifumi Uesono

Molecular Pharmacology October 5, 2018, mol.118.112656; DOI: https://doi.org/10.1124/mol.118.112656
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Activated CaMKIIα binds to the mGlu5 metabotropic glutamate receptor and modulates calcium mobilization
Christian R Marks, Brian C Shonesy, Xiaohan Wang, Jason R Stephenson, Colleen Niswender and Roger J Colbran

Molecular Pharmacology October 3, 2018, mol.118.113142; DOI: https://doi.org/10.1124/mol.118.113142
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Reduced Activity of GGPPS Mutant is Involved in Bisphosphonates-Induced Atypical Fractures
Michal Lisnyansky, Noa Kapelushnik, Ariel Ben-Bassat, Milit Marom, Anat Loewenstein, Daniel Khananshvili, Moshe Giladi and Yoni Haitin

Molecular Pharmacology October 1, 2018, mol.118.113670; DOI: https://doi.org/10.1124/mol.118.113670
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Functional Expression of Organic Anion Transporting Polypeptide 1a4 (Oatp1a4) is Regulated by Transforming Growth Factor-/Activin Receptor-like Kinase 1 (TGF-/ALK1) Signaling at the Blood-Brain Barrier
Wazir Abdullahi, Hrvoje Brzica, Nicholas A. Hirsch, Bianca G. Reilly and Patrick T. Ronaldson

Molecular Pharmacology September 27, 2018, mol.118.112912; DOI: https://doi.org/10.1124/mol.118.112912
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Differential effects of integrin αv knockdown and cilengitide on sensitisation of triple-negative breast cancer and melanoma cells to microtubule poisons
Nikolina Stojanovic, Ana Dekanic, Mladen Paradzik, Dragomira Majhen, Kresimir Ferencak, Jelena Ruscic, Irena Bardak, Christine Supina, Maja T. Tomicic, Markus Christmann, Maja Osmak and Andreja Ambriovic-Ristov

Molecular Pharmacology September 27, 2018, mol.118.113027; DOI: https://doi.org/10.1124/mol.118.113027
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Modeling and mutational analysis of the binding mode for the multimodal antidepressant drug vortioxetine to the human 5-HT3A receptor
Lucy Kate Ladefoged, Lachlan Munro, Anders J Pedersen, Thomas Balle, Benny Bang-Andersen, Sarah C R Lummis, Birgit Schiott and Anders S Kristensen

Molecular Pharmacology September 26, 2018, mol.118.113530; DOI: https://doi.org/10.1124/mol.118.113530
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Homogeneous, real-time NanoBRET binding assays for the histamine H₃ and H₄ receptor on living cells
Tamara A.M. Mocking, Eleonore W.E. Verweij, Henry F Vischer and Rob Leurs

Molecular Pharmacology September 24, 2018, mol.118.113373; DOI: https://doi.org/10.1124/mol.118.113373
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Betacellulin (BTC) Biases the EGFR to Dimerize with ErbB3
Jamie S Rush, Joanne L Peterson and Brian P Ceresa

Molecular Pharmacology September 24, 2018, mol.118.113399; DOI: https://doi.org/10.1124/mol.118.113399

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APPLYING THE MONOD-WYMAN-CHANGEUX ALLOSTERIC ACTIVATION MODEL TO PSEUDO-STEADY-STATE RESPONSES FROM GABAA RECEPTORS
Joseph H. Steinbach and Gustav Akk

Molecular Pharmacology October 17, 2018, mol.118.113787; DOI: https://doi.org/10.1124/mol.118.113787

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