Fast Forward

Molecular Pharmacology Fast Forward contains papers in manuscript form that have been accepted and published in Molecular Pharmacology but have not been copyedited and have not been assigned to an issue of the journal. Copyediting may lead to some differences between the Fast Forward version and the final version. There may also be differences in the quality of the graphics. The publication date appears below each title followed by the article's unique Digital Object Identifier (DOI).

Articles

You have access
Non-classical ligand-independent regulation of Go protein by an orphan Class C GPCR
Mariana Hajj, Teresa De Vita, Claire Vol, Charlotte Renassia, Jean-Charles Bologna, Isabelle Brabet, Magali Cazade, Manuela Pastore, Jaroslav Blahos, Gilles Labesse, Jean-Philippe Pin and Laurent Prezeau

Molecular Pharmacology June 12, 2019, mol.118.113019; DOI: https://doi.org/10.1124/mol.118.113019
You have access
Generation and characterization of an Abcc1 humanized mouse model (hABCC1flx/flx) with knockout capability
Markus Krohn, Victoria Zoufal, Severin Mairinger, Thomas Wanek, Kristin Paarmann, Thomas Bruning, Ivan Eiriz, Mirjam Brackhan, Oliver Langer and Jens Pahnke

Molecular Pharmacology June 12, 2019, mol.119.115824; DOI: https://doi.org/10.1124/mol.119.115824
You have access
Identification of Serine-875 as an Inhibitory Phosphorylation Site in the Calcium-Sensing Receptor
Lenah S Binmahfouz, Patricia P Centeno, Arthur D Conigrave and Donald T Ward

Molecular Pharmacology June 12, 2019, mol.119.116178; DOI: https://doi.org/10.1124/mol.119.116178
You have access
The Pore-Lipid Interface: Role of Amino Acid Determinants of Lipophilic Access by Ivabradine to the hERG1 Pore Domain
Henry J Duff, Sergei Y Noskov, Danielle Muruve, German Perlovic, Marina Ol Khovich, Angelica Sharapova, Brenda Gerull, Jiqing Guo, Meryuvert Kudaibergenova and Laura Perissinotti

Molecular Pharmacology June 10, 2019, mol.118.115642; DOI: https://doi.org/10.1124/mol.118.115642
You have access
Severe Hepatotoxicity of Mithramycin Therapy Caused by Altering Expression of Hepatocellular Bile Transporters
Tristan M. Sissung, Phoebe A. Huang, Ralph J Hauke, Edel M. McCrea, Cody J. Peer, Roberto H. Barbier, Jonathan D. Strope, Ariel M. Ley, Mary Zhang, Julie A. Hong, David Venzon, Jonathan P. Jackson, Kenneth R. Brouwer, Patrick Grohar, Jon Glod, Brigitte C. Widemann, Theo Heller, David S. Schrump and William D Figg

Molecular Pharmacology June 7, 2019, mol.118.114827; DOI: https://doi.org/10.1124/mol.118.114827
You have access
The L46P mutant confers a novel allosteric mechanism of resistance towards the influenza A virus M2 S31N proton channel blockers
Rami Musharrafieh, Panagiotis Lagarias, Chunlong Ma, Gene Tan, Antonios Kolocouris and Jun Wang

Molecular Pharmacology June 7, 2019, mol.119.116640; DOI: https://doi.org/10.1124/mol.119.116640
You have access
Investigating the Binding Interactions of NS6740, a Silent Agonist of the Nicotinic Receptor
Catriona E. W. Blunt and Dennis A. Dougherty

Molecular Pharmacology June 7, 2019, mol.119.116244; DOI: https://doi.org/10.1124/mol.119.116244
You have access
Inhibition of Heat shock protein 90 suppresses Twist1 transcription
Kay Yi Chong, Min Kang, Francesca Garofalo, Daiki Ueno, Huamao Liang, Sarah Cady, Oluwagbemisola Madarikan, Nicholas Pitruzzello, Cheng-Hsiu Tsai, Tobias Hartwich, Brian Shuch and Yang Yang-Hartwich

Molecular Pharmacology June 7, 2019, mol.119.116137; DOI: https://doi.org/10.1124/mol.119.116137
You have access
Modulation of burst firing of neurons in nucleus reticularis of the thalamus by GluN2C-containing NMDA receptors
Jinxu Liu, Gajanan P Shelkar, Fabao Zhao, Rasmus Praetorius Clausen and Shashank Manohar Dravid

Molecular Pharmacology June 3, 2019, mol.119.116780; DOI: https://doi.org/10.1124/mol.119.116780
You have access
Evidence for the Interaction of A₃ Adenosine Receptor Agonists at the Drug-Binding Site(s) of Human P-glycoprotein (ABCB1)
Biebele Abel, Dilip K. Tosh, Stewart R. Durell, Megumi Murakami, Shahrooz Vahedi, Kenneth A. Jacobson and Suresh V. Ambudkar

Molecular Pharmacology May 24, 2019, mol.118.115295; DOI: https://doi.org/10.1124/mol.118.115295
You have access
OATP1B3-1B7 (LST-3TM12) is a drug transporter that affects endoplasmic reticulum access and the metabolism of ezetimibe
Vanessa Malagnino, Urs Duthaler, Isabell Seibert, Stephan Krahenbuhl and Henriette Elisabeth Meyer zu Schwabedissen

Molecular Pharmacology May 24, 2019, mol.118.114934; DOI: https://doi.org/10.1124/mol.118.114934

Minireview

You have access
A biased view of µ opioid receptors?
Alexandra E Conibear and Eamonn Kelly

Molecular Pharmacology June 7, 2019, mol.119.115956; DOI: https://doi.org/10.1124/mol.119.115956
You have access
Insights into Doxorubicin-induced Cardiotoxicity: Molecular Mechanisms, Preventive Strategies, and Early Monitoring
Nadine Wenningmann, Merle Knapp, Anusha Ande, Tanaya R Vaidya and Sihem Ait-Oudhia

Molecular Pharmacology June 4, 2019, mol.119.115725; DOI: https://doi.org/10.1124/mol.119.115725
You have access
Context-dependent signalling of CXC chemokine receptor 4 (CXCR4) and atypical chemokine receptor 3 (ACKR3)
Joyce Heuninck, Cristina Perpina Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J Briddon, Thierry Durroux, Stephen J Hill, Martin J Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten Hoffmann

Molecular Pharmacology May 15, 2019, mol.118.115477; DOI: https://doi.org/10.1124/mol.118.115477
You have access
Atypical chemokine receptor 3 (ACKR3): a comprehensive overview of its expression and potential roles in the immune system.
Joyce Koenen, Francoise Bachelerie, Karl Balabanian, Geraldine Schlecht-Louf and Carmen Gallego

Molecular Pharmacology April 30, 2019, mol.118.115329; DOI: https://doi.org/10.1124/mol.118.115329
You have access
Does the lipid bilayer orchestrate access and binding of ligands to transmembrane orthosteric/allosteric sites of GPCRs?
Christopher Tytus Szlenk, Jeevan B GC and Senthil Natesan

Molecular Pharmacology April 8, 2019, mol.118.115113; DOI: https://doi.org/10.1124/mol.118.115113
You have access
CXCR4/ACKR3 phosphorylation and recruitment of interacting proteins: key mechanisms regulating their functional status
Amos Fumagalli, Aurelien Zarca, Maria Neves, Birgit Caspar, Stephen J Hill, Federico Mayor, Martine J Smit and Philippe Marin

Molecular Pharmacology March 5, 2019, mol.118.115360; DOI: https://doi.org/10.1124/mol.118.115360
You have access
The role of ACKR3 in breast, lung and brain cancer.
Maria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J Smit and Federico Mayor

Molecular Pharmacology February 11, 2019, mol.118.115279; DOI: https://doi.org/10.1124/mol.118.115279

Main menu

User menu

Search

Fast Forward

Articles

Minireview

Navigate

More Information

ASPET's Other Journals