Table of Contents

Articles

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  Colorectal Cancer-Specific Cytochrome P450 2W1: Intracellular Localization, Glycosylation, and Catalytic Activity

  Alvin Gomez, Jana Nekvindova, Sandra Travica, Mi-Young Lee, Inger Johansson, David Edler, Souren Mkrtchian and Magnus Ingelman-Sundberg

  Molecular Pharmacology December 2010, 78 (6) 1004-1011; DOI: https://doi.org/10.1124/mol.110.067652
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  Tethered Agonist Analogs as Site-Specific Probes for Domains of the Human α7 Nicotinic Acetylcholine Receptor that Differentially Regulate Activation and Desensitization

  Jingyi Wang, Nicole A. Horenstein, Clare Stokes and Roger L. Papke

  Molecular Pharmacology December 2010, 78 (6) 1012-1025; DOI: https://doi.org/10.1124/mol.110.066662
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  The High-Affinity Binding Site for Tricyclic Antidepressants Resides in the Outer Vestibule of the Serotonin Transporter

  Subhodeep Sarker, René Weissensteiner, Ilka Steiner, Harald H. Sitte, Gerhard F. Ecker, Michael Freissmuth and Sonja Sucic

  Molecular Pharmacology December 2010, 78 (6) 1026-1035; DOI: https://doi.org/10.1124/mol.110.067538
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  Mapping the Ligand Binding Sites of Kainate Receptors: Molecular Determinants of Subunit-Selective Binding of the Antagonist [³H]UBP310

  Palmi T. Atlason, Caroline L. Scholefield, Richard J. Eaves, M. Belen Mayo-Martin, David E. Jane and Elek Molnár

  Molecular Pharmacology December 2010, 78 (6) 1036-1045; DOI: https://doi.org/10.1124/mol.110.067934
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  Identification of 5α,6α-Epoxycholesterol as a Novel Modulator of Liver X Receptor Activity

  Thomas J. Berrodin, Qi Shen, Elaine M. Quinet, Matthew R. Yudt, Leonard P. Freedman and Sunil Nagpal

  Molecular Pharmacology December 2010, 78 (6) 1046-1058; DOI: https://doi.org/10.1124/mol.110.065193
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  ATP Induces Synaptic Gene Expressions in Cortical Neurons: Transduction and Transcription Control via P2Y₁ Receptors

  Nina L. Siow, Roy C. Y. Choi, Heidi Q. Xie, Ling W. Kong, Glanice K. Y. Chu, Gallant K. L. Chan, Joseph Simon, Eric A. Barnard and Karl W. K. Tsim

  Molecular Pharmacology December 2010, 78 (6) 1059-1071; DOI: https://doi.org/10.1124/mol.110.066506
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  Emetine Promotes von Hippel-Lindau-Independent Degradation of Hypoxia-Inducible Factor-2α in Clear Cell Renal Carcinoma

  Hye-Sik Kong, Sunmin Lee, Kristin Beebe, Bradley Scroggins, Gopal Gupta, Min-Jung Lee, Yun-Jin Jung, Jane Trepel and Leonard Neckers

  Molecular Pharmacology December 2010, 78 (6) 1072-1078; DOI: https://doi.org/10.1124/mol.110.066514
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  The Human Organic Anion Transporter Genes OAT5 and OAT7 Are Transactivated by Hepatocyte Nuclear Factor-1α (HNF-1α)

  Kerstin Klein, Christoph Jüngst, Jessica Mwinyi, Bruno Stieger, Franz Krempler, Wolfgang Patsch, Jyrki J. Eloranta and Gerd A. Kullak-Ublick

  Molecular Pharmacology December 2010, 78 (6) 1079-1087; DOI: https://doi.org/10.1124/mol.110.065201
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  The Specific Slow Afterhyperpolarization Inhibitor UCL2077 Is a Subtype-Selective Blocker of the Epilepsy Associated KCNQ Channels

  Heun Soh and Anastassios V. Tzingounis

  Molecular Pharmacology December 2010, 78 (6) 1088-1095; DOI: https://doi.org/10.1124/mol.110.066100
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  Melanoma Differentiation Associated Gene-7/Interleukin-24 Potently Induces Apoptosis in Human Myeloid Leukemia Cells through a Process Regulated by Endoplasmic Reticulum Stress

  Mohamed Rahmani, Mandy Mayo, Rupesh Dash, Upneet Kaur Sokhi, Igor P. Dmitriev, Devanand Sarkar, Paul Dent, David T. Curiel, Paul B. Fisher and Steven Grant

  Molecular Pharmacology December 2010, 78 (6) 1096-1104; DOI: https://doi.org/10.1124/mol.110.068007
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  Discovery of Novel Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5 Reveals Chemical and Functional Diversity and In Vivo Activity in Rat Behavioral Models of Anxiolytic and Antipsychotic Activity

  Alice L. Rodriguez, Mark D. Grier, Carrie K. Jones, Elizabeth J. Herman, Alexander S. Kane, Randy L. Smith, Richard Williams, Ya Zhou, Joy E. Marlo, Emily L. Days, Tasha N. Blatt, Satyawan Jadhav, Usha N. Menon, Paige N. Vinson, Jerri M. Rook, Shaun R. Stauffer, Colleen M. Niswender, Craig W. Lindsley, C. David Weaver and P. Jeffrey Conn

  Molecular Pharmacology December 2010, 78 (6) 1105-1123; DOI: https://doi.org/10.1124/mol.110.067207
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  The Tarantula Toxins ProTx-II and Huwentoxin-IV Differentially Interact with Human Na_v1.7 Voltage Sensors to Inhibit Channel Activation and Inactivation

  Yucheng Xiao, Kenneth Blumenthal, James O. Jackson, Songping Liang and Theodore R. Cummins

  Molecular Pharmacology December 2010, 78 (6) 1124-1134; DOI: https://doi.org/10.1124/mol.110.066332