Index by author

September 01, 2013; Volume 84,Issue 3

A

  1. Ahmed, M. Shakil

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  2. Alpizar, Yeranddy A.

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  3. Ambudkar, Suresh V.

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

  4. Appel, Jon R.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  5. Attramadal, Håvard

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

B

  1. Baker, Daniel L.

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  2. Bittman, Robert

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  3. Boonen, Brett

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

C

  1. Cheepala, Satish B.

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

  2. Christopoulos, Arthur

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  3. Corrêa, Ivan R.

    1. Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
      Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
      Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868

  4. Crooks, Peter A.

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

D

  1. Devine, Shane M.

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  2. Dragin, Nadine

    1. Oral Benzo[a]pyrene: Understanding Pharmacokinetics, Detoxication, and Consequences—Cyp1 Knockout Mouse Lines as a Paradigm
      Daniel W. Nebert, Zhanquan Shi, Marina Gálvez-Peralta, Shigeyuki Uno and Nadine Dragin
      Molecular Pharmacology September 2013, 84 (3) 304-313; DOI: https://doi.org/10.1124/mol.113.086637

  3. Drenan, Ryan M.

    1. α4α6β2* Nicotinic Acetylcholine Receptor Activation on Ventral Tegmental Area Dopamine Neurons Is Sufficient to Stimulate a Depolarizing Conductance and Enhance Surface AMPA Receptor Function
      Staci E. Engle, Pei-Yu Shih, J. Michael McIntosh and Ryan M. Drenan
      Molecular Pharmacology September 2013, 84 (3) 393-406; DOI: https://doi.org/10.1124/mol.113.087346

E

  1. Edvardsen, Thor

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  2. Edwards, Bruce S.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  3. Ehrlich, Aliza T.

    1. Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing Gβγ Subunits in Human Embryonic Kidney 293T Cells
      Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya
      Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288

  4. Ekins, Sean

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

  5. Engle, Staci E.

    1. α4α6β2* Nicotinic Acetylcholine Receptor Activation on Ventral Tegmental Area Dopamine Neurons Is Sufficient to Stimulate a Depolarizing Conductance and Enhance Surface AMPA Receptor Function
      Staci E. Engle, Pei-Yu Shih, J. Michael McIntosh and Ryan M. Drenan
      Molecular Pharmacology September 2013, 84 (3) 393-406; DOI: https://doi.org/10.1124/mol.113.087346

  6. Everaerts, Wouter

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  7. Everett, Steven

    1. Specificity Determinants of CYP1B1 Estradiol Hydroxylation
      Clinton R. Nishida, Steven Everett and Paul R. Ortiz de Montellano
      Molecular Pharmacology September 2013, 84 (3) 451-458; DOI: https://doi.org/10.1124/mol.113.087700

F

  1. Fells, James I.

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  2. Fifer, E. Kim

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

  3. Fujiwara, Yuko

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  4. Fukuda, Yu

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

  5. Furuyashiki, Tomoyuki

    1. Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing Gβγ Subunits in Human Embryonic Kidney 293T Cells
      Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya
      Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288

G

  1. Gálvez-Peralta, Marina

    1. Oral Benzo[a]pyrene: Understanding Pharmacokinetics, Detoxication, and Consequences—Cyp1 Knockout Mouse Lines as a Paradigm
      Daniel W. Nebert, Zhanquan Shi, Marina Gálvez-Peralta, Shigeyuki Uno and Nadine Dragin
      Molecular Pharmacology September 2013, 84 (3) 304-313; DOI: https://doi.org/10.1124/mol.113.086637

  2. Gavalas, Anthony

    1. Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
      Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
      Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868

  3. Gees, Maarten

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  4. Giulianotti, Marc A.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  5. Gorren, Antonius C. F.

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  6. Gravning, Jørgen

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

H

  1. Hagelin, Else Marie V.

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  2. Hals, Petter-Arnt

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

  3. Hansen, Lærke S.

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  4. Hascher, Antje

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

  5. Heideman, Warren

    1. Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish
      Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman
      Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413

  6. Hofsteen, Peter

    1. Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish
      Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman
      Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413

  7. Houghten, Richard A.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  8. Hummel-Eisenbeiss, Johanna

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

J

  1. Janssens, Annelies

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  2. Javitch, Jonathan A.

    1. Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
      Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
      Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868

  3. Johnson, Shaina D.

    1. Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish
      Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman
      Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413

K

  1. Kakizuka, Akira

    1. Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing Gβγ Subunits in Human Embryonic Kidney 293T Cells
      Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya
      Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288

  2. Keov, Peter

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  3. Kimbrell, Matthew R.

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

  4. Kirby, R. Jason

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  5. Kitaoka, Shiho

    1. Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing Gβγ Subunits in Human Embryonic Kidney 293T Cells
      Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya
      Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288

  6. Koesling, Doris

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  7. Krobert, Kurt

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

L

  1. Lambert, Nevin A.

    1. Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
      Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
      Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868

  2. Lan, Tien-Hung

    1. Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
      Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
      Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868

  3. Lane, J. Robert

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  4. Lang, Barbara

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  5. Lee, Sue Chin

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  6. Levy, Finn Olav

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  7. Lim, Keng Gat

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  8. Liu, Jianxiong

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  9. Liu, Qiuju

    1. Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
      Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
      Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868

  10. Lyko, Frank

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

M

  1. Mayer, Bernd

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  2. McIntosh, J. Michael

    1. α4α6β2* Nicotinic Acetylcholine Receptor Activation on Ventral Tegmental Area Dopamine Neurons Is Sufficient to Stimulate a Depolarizing Conductance and Enhance Surface AMPA Receptor Function
      Staci E. Engle, Pei-Yu Shih, J. Michael McIntosh and Ryan M. Drenan
      Molecular Pharmacology September 2013, 84 (3) 393-406; DOI: https://doi.org/10.1124/mol.113.087346

  3. Medina-Franco, Jose L.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  4. Miller, Duane D.

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  5. Moe, Ingvild Tronstad

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  6. Müller-Tidow, Carsten

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

N

  1. Namkung, Wan

    1. Novel Amino-Carbonitrile-Pyrazole Identified in a Small Molecule Screen Activates Wild-Type and ∆F508 Cystic Fibrosis Transmembrane Conductance Regulator in the Absence of a cAMP Agonist
      Wan Namkung, Jinhong Park, Yohan Seo and A. S. Verkman
      Molecular Pharmacology September 2013, 84 (3) 384-392; DOI: https://doi.org/10.1124/mol.113.086348

  2. Narumiya, Shuh

    1. Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing Gβγ Subunits in Human Embryonic Kidney 293T Cells
      Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya
      Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288

  3. Nebert, Daniel W.

    1. Oral Benzo[a]pyrene: Understanding Pharmacokinetics, Detoxication, and Consequences—Cyp1 Knockout Mouse Lines as a Paradigm
      Daniel W. Nebert, Zhanquan Shi, Marina Gálvez-Peralta, Shigeyuki Uno and Nadine Dragin
      Molecular Pharmacology September 2013, 84 (3) 304-313; DOI: https://doi.org/10.1124/mol.113.086637

  4. Nelson, Sandra

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  5. Neubauer, Andrea

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  6. Neubauer, Regina

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  7. Nilius, Bernd

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  8. Nishida, Clinton R.

    1. Specificity Determinants of CYP1B1 Estradiol Hydroxylation
      Clinton R. Nishida, Steven Everett and Paul R. Ortiz de Montellano
      Molecular Pharmacology September 2013, 84 (3) 451-458; DOI: https://doi.org/10.1124/mol.113.087700

  9. Norman, Derek D.

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

O

  1. Ortiz de Montellano, Paul R.

    1. Specificity Determinants of CYP1B1 Estradiol Hydroxylation
      Clinton R. Nishida, Steven Everett and Paul R. Ortiz de Montellano
      Molecular Pharmacology September 2013, 84 (3) 451-458; DOI: https://doi.org/10.1124/mol.113.087700

  2. Osnes, Jan-Bjørn

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  3. Owsianik, Grzegorz

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

P

  1. Pack, Thomas F.

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

  2. Papke, Roger L.

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

  3. Papoian, Ruben

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  4. Park, Jinhong

    1. Novel Amino-Carbonitrile-Pyrazole Identified in a Small Molecule Screen Activates Wild-Type and ∆F508 Cystic Fibrosis Transmembrane Conductance Regulator in the Absence of a cAMP Agonist
      Wan Namkung, Jinhong Park, Yohan Seo and A. S. Verkman
      Molecular Pharmacology September 2013, 84 (3) 384-392; DOI: https://doi.org/10.1124/mol.113.086348

  5. Parrill, Abby L.

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  6. Patil, Renukadevi

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  7. Peng, Can

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

  8. Petersen, Trine P.

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  9. Peterson, Richard E.

    1. Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish
      Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman
      Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413

  10. Pinilla, Clemencia

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  11. Plavicki, Jessica

    1. Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish
      Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman
      Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413

Q

  1. Qvigstad, Eirik

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

R

  1. Rius, Maria

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

  2. Rosenkilde, Mette M.

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  3. Rummel, Pia C.

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  4. Russwurm, Michael

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

S

  1. Sagave, Julia

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  2. Sanchez, Alicia

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  3. Sandvold, Marit Liland

    1. The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
      Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
      Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801

  4. Santos, Radleigh G.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  5. Scammells, Peter J.

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  6. Schmidt, Kurt

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  7. Schrammel, Astrid

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  8. Schuetz, John D.

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

  9. Schwarzenegger, Christine

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  10. Segal, Andrei

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  11. Seibel, William

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  12. Seo, Yohan

    1. Novel Amino-Carbonitrile-Pyrazole Identified in a Small Molecule Screen Activates Wild-Type and ∆F508 Cystic Fibrosis Transmembrane Conductance Regulator in the Absence of a cAMP Agonist
      Wan Namkung, Jinhong Park, Yohan Seo and A. S. Verkman
      Molecular Pharmacology September 2013, 84 (3) 384-392; DOI: https://doi.org/10.1124/mol.113.086348

  13. Sexton, Patrick M.

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  14. Shi, Zhanquan

    1. Oral Benzo[a]pyrene: Understanding Pharmacokinetics, Detoxication, and Consequences—Cyp1 Knockout Mouse Lines as a Paradigm
      Daniel W. Nebert, Zhanquan Shi, Marina Gálvez-Peralta, Shigeyuki Uno and Nadine Dragin
      Molecular Pharmacology September 2013, 84 (3) 304-313; DOI: https://doi.org/10.1124/mol.113.086637

  15. Shih, Pei-Yu

    1. α4α6β2* Nicotinic Acetylcholine Receptor Activation on Ventral Tegmental Area Dopamine Neurons Is Sufficient to Stimulate a Depolarizing Conductance and Enhance Surface AMPA Receptor Function
      Staci E. Engle, Pei-Yu Shih, J. Michael McIntosh and Ryan M. Drenan
      Molecular Pharmacology September 2013, 84 (3) 393-406; DOI: https://doi.org/10.1124/mol.113.087346

  16. Sklar, Larry A.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  17. Skomedal, Tor

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  18. Sparre-Ulrich, Alexander H.

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  19. Sparreboom, Alex

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

T

  1. Takenaka, Kazumasa

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

  2. Talavera, Karel

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

  3. Thiele, Stefanie

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  4. Tian, Chengju

    1. Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
      Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
      Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462

  5. Tigyi, Gabor

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

  6. Tsukahara, Ryoko

    1. Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
      James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
      Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080

U

  1. Ulven, Trond

    1. Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
      Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
      Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702

  2. Uno, Shigeyuki

    1. Oral Benzo[a]pyrene: Understanding Pharmacokinetics, Detoxication, and Consequences—Cyp1 Knockout Mouse Lines as a Paradigm
      Daniel W. Nebert, Zhanquan Shi, Marina Gálvez-Peralta, Shigeyuki Uno and Nadine Dragin
      Molecular Pharmacology September 2013, 84 (3) 304-313; DOI: https://doi.org/10.1124/mol.113.086637

V

  1. Valant, Celine

    1. Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
      Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
      Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320

  2. Valen, Guro

    1. Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
      Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
      Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312

  3. Verkman, A. S.

    1. Novel Amino-Carbonitrile-Pyrazole Identified in a Small Molecule Screen Activates Wild-Type and ∆F508 Cystic Fibrosis Transmembrane Conductance Regulator in the Absence of a cAMP Agonist
      Wan Namkung, Jinhong Park, Yohan Seo and A. S. Verkman
      Molecular Pharmacology September 2013, 84 (3) 384-392; DOI: https://doi.org/10.1124/mol.113.086348

  4. Voets, Thomas

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

W

  1. Wölkart, Gerald

    1. Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
      Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
      Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835

  2. Wu, Chung-Pu

    1. Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
      Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
      Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967

X

  1. Xue, Fenqin

    1. Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
      Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
      Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548

Y

  1. Yates-Gibbins, Tina

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595

  2. Young, Susan M.

    1. Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
      Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
      Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595
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