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Molecular Basis of Metabolism-Mediated Conversion of PK11195 from an Antagonist to an Agonist of the Constitutive Androstane Receptor

Bryan Mackowiak, Linhao Li, Matthew A. Welch, Daochuan Li, Jace W. Jones, Scott Heyward, Maureen A. Kane, Peter W. Swaan and Hongbing Wang
Molecular Pharmacology July 2017, 92 (1) 75-87; DOI: https://doi.org/10.1124/mol.117.108621
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Research ArticleArticle

Metabolism-Based Antagonism/Agonism Conversion of PK11195

Bryan Mackowiak, Linhao Li, Matthew A. Welch, Daochuan Li, Jace W. Jones, Scott Heyward, Maureen A. Kane, Peter W. Swaan and Hongbing Wang
Molecular Pharmacology July 1, 2017, 92 (1) 75-87; DOI: https://doi.org/10.1124/mol.117.108621
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